Name Target Type Structure Assay KD (uM) cellular CD47/SIRPα IC50 (uM) Citation
pep-20 CD47 linear peptide AWSATWSNYWRH MST 3.2 ± 2.3 25 10.1136/jitc-2020-000905
pep-3 CD47 linear peptide TDLRYKEHYLYL MST 0.7 ± 4.6 NA 10.1136/jitc-2020-000905
pep-20-D12 CD47 linear peptide a w s ATWSNY w r h FC CD47-SIRPα competition NA 12 10.1136/jitc-2020-000905
RS-17 CD47 linear peptide RRYKQDGGWSHWSPPWSS MST 0.004 ± 0.001 NA CN110981942
D4-1 SIRPα cyclicpeptide Ac*-yKDWSISARITPVHPCG-NH2 SPR 0.012 NA 10.1016/j.chembiol.2020.06.008
D4-2 SIRPα cyclicpeptide Ac*-yRYSAVYSIHPSWC*G-NH2 SPR 0.011 0.18 10.1016/j.chembiol.2020.06.008
L4-4 SIRPα cyclicpeptide Ac*-YYALSDRYTALYPKPC*G-NH2 SPR 0.006 NA 10.1016/j.chembiol.2020.06.008
SP5 SIRPα cyclicpeptide C*TQDAWHIC* MST 0.38 NA CN111116713